Compile Data Set for Download or QSAR
maximum 50k data
Found 36 of ic50 data for polymerid = 50003371,50005949,50006462
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM14673(Fragment 3 | Malonic Acid | propanedioic acid)
Affinity DataIC50:  2.49E+4nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50038343(CHEMBL3360546)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibition of mouse serine racemase using L-serine substrate by reversed-phase HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM14673(Fragment 3 | Malonic Acid | propanedioic acid)
Affinity DataIC50:  6.70E+4nMAssay Description:Inhibition of mouse serine racemase using L-serine substrate by reversed-phase HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378531(CHEMBL566071)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of mouse recombinant serine racemase expressed in Escherichia coli MC1061 assessed as formation of D-serine after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50038354(CHEBI:16513 | CHEMBL1794676)
Affinity DataIC50:  9.40E+4nMAssay Description:Inhibition of mouse serine racemase using L-serine substrate by reversed-phase HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM31147(4H-furo[3,2-b]pyrrole-5-carboxylic acid | 5-carbox...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50055464(CHEMBL3317747)
Affinity DataIC50:  1.40E+5nMAssay Description:Inhibition of serine racemase mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378530(CHEMBL566494)
Affinity DataIC50:  1.70E+5nMAssay Description:Inhibition of mouse recombinant serine racemase expressed in Escherichia coli MC1061 assessed as formation of D-serine after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378532(CHEMBL569435)
Affinity DataIC50:  3.70E+5nMAssay Description:Inhibition of mouse recombinant serine racemase expressed in Escherichia coli MC1061 assessed as formation of D-serine after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM92990(Aminomalonate)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibition of mouse serine racemase using L-serine substrate by reversed-phase HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50055465(CHEMBL3317754)
Affinity DataIC50:  5.20E+5nMAssay Description:Inhibition of full length human recombinant serine recemase C2DC6D mutant expressed in Escherichia coli BL21 (DE3) assessed as D-serine production af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50055466(CHEMBL3317759)
Affinity DataIC50:  6.30E+5nMAssay Description:Inhibition of full length human recombinant serine recemase C2DC6D mutant expressed in Escherichia coli BL21 (DE3) assessed as D-serine production af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50038342(CHEMBL3360547)
Affinity DataIC50:  7.80E+5nMAssay Description:Inhibition of mouse serine racemase using L-serine substrate by reversed-phase HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50453342(CHEMBL4205674)
Affinity DataIC50:  8.36E+5nMAssay Description:Inhibition of wild-type serine racemase (unknown origin) assessed as residual activity by measuring D-serine level using Dsd1 as substrate and PLP as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50055464(CHEMBL3317747)
Affinity DataIC50:  1.21E+6nMAssay Description:Inhibition of full length human recombinant serine recemase C2DC6D mutant expressed in Escherichia coli BL21 (DE3) assessed as D-serine production af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50129194((2S)-2-amino-4-(hydroxyamino)-4-oxobutanoic acidN(...)
Affinity DataIC50:  1.30E+6nMAssay Description:Inhibition of mouse recombinant serine racemase expressed in Escherichia coli MC1061 assessed as formation of D-serine after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM14673(Fragment 3 | Malonic Acid | propanedioic acid)
Affinity DataIC50:  1.31E+6nMAssay Description:Inhibition of full length human recombinant serine recemase C2DC6D mutant expressed in Escherichia coli BL21 (DE3) assessed as D-serine production af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50055464(CHEMBL3317747)
Affinity DataIC50:  1.60E+6nMAssay Description:Inhibition of wild-type serine racemase (unknown origin) assessed as residual activity by measuring D-serine level using Dsd1 as substrate and PLP as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50038341(CHEBI:30860 | METHYLMALONIC ACID)
Affinity DataIC50:  1.85E+6nMAssay Description:Inhibition of mouse serine racemase using L-serine substrate by reversed-phase HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50038340(CHEMBL3360548)
Affinity DataIC50:  2.16E+6nMAssay Description:Inhibition of mouse serine racemase using L-serine substrate by reversed-phase HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427212((2S,3R)-2,3-Dihydroxysuccinic Acid | CHEMBL225983 ...)
Affinity DataIC50:  2.82E+6nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427205(CHEMBL2324854)
Affinity DataIC50: >5.00E+6nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427209(CHEMBL1497209)
Affinity DataIC50:  5.02E+6nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427211(CHEMBL2324857)
Affinity DataIC50:  5.16E+6nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427206(CHEMBL2324852)
Affinity DataIC50:  5.28E+6nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50038339(CHEMBL3360549)
Affinity DataIC50:  5.63E+6nMAssay Description:Inhibition of mouse serine racemase using L-serine substrate by reversed-phase HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427210(CHEMBL2324858)
Affinity DataIC50:  5.72E+6nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50038338(CHEMBL3360550)
Affinity DataIC50:  7.03E+6nMAssay Description:Inhibition of mouse serine racemase using L-serine substrate by reversed-phase HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50074328(CHEMBL164585 | Thiophene-3-carboxylic acid)
Affinity DataIC50:  8.21E+6nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50146456((2E)-3-(3-hydroxyphenyl)-2-propenoic acid | (2E)-3...)
Affinity DataIC50:  8.39E+6nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427207(CROTONIC ACID | Crotonate)
Affinity DataIC50: >1.00E+7nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM36181(SODIUM BENZOATE | benzoate | benzoic acid | benzoi...)
Affinity DataIC50: >1.00E+7nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427204(CHEMBL2324856)
Affinity DataIC50: >1.00E+7nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50206007(3-Hydroxy-chromen-2-one | 3-hydroxy-2H-chromen-2-o...)
Affinity DataIC50: >1.00E+7nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427208(CHEMBL554820)
Affinity DataIC50: >1.00E+7nMAssay Description:Inhibition of human recombinant N-terminal His-tagged serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate after 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Mus musculus)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50038355(CHEMBL3360551)
Affinity DataIC50:  4.06E+7nMAssay Description:Inhibition of mouse serine racemase using L-serine substrate by reversed-phase HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed